Literature Box
Help
SEARCH
PI, Family, Clan or Protein ID
Authors
Title
Year
Category
type code
Advanced search Clear

PI, Family, Clan or Protein ID Authors Title Source Year PubMed DOI Category
I12.002 Legowska,A., Debowski,D., Lesner,A., Wysocka,M. & Rolka,K. Selection of peptomeric inhibitors of bovine alpha-chymotrypsin and cathepsin G based on trypsin inhibitor SFTI-1 using a combinatorial chemistry approach Mol Divers (2010) 14, 51-58. 2010 PubMed DOI Design of small-molecule Inhibitors
I12.002 Pereira,H.J., Salgado,M.C. & Oliveira,E.B. Immobilized analogues of sunflower trypsin inhibitor-1 constitute a versatile group of affinity sorbents for selective isolation of serine proteases J Chromatogr B Analyt Technol Biomed Life Sci (2009) 877, 2039-2044. 2009 PubMed DOI
I12.002 Legowska,A., Debowski,D., Lesner,A., Wysocka,M. & Rolka,K. Introduction of non-natural amino acid residues into the substrate-specific P1 position of trypsin inhibitor SFTI-1 yields potent chymotrypsin and cathepsin G inhibitors Bioorg Med Chem (2009) 17, 3302-3307. 2009 PubMed DOI Mutation, allelic variant or polymorphism
I12.002 Garcia Boy,R., Mier,W., Nothelfer,E.M., Altmann,A., Eisenhut,M., Kolmar,H., Tomaszowski,M., Kramer,S. & Haberkorn,U. Sunflower trypsin inhibitor 1 derivatives as molecular scaffolds for the development of novel peptidic radiopharmaceuticals Mol Imaging Biol (2009) 2009 PubMed DOI Suggested therapeutcal potential
I12.002 Legowska,A., Bulak,E., Wysocka,M., Jaskiewicz,A., Lesner,A., Debowski,D. & Rolka,K. Peptomeric analogues of trypsin inhibitor SFTI-1 isolated from sunflower seeds Bioorg Med Chem (2008) 16, 5644-5652. 2008 PubMed DOI Design of small-molecule Inhibitors
I12.002 Li,P., Jiang,S., Lee,S.L., Lin,C.Y., Johnson,M.D., Dickson,R.B., Michejda,C.J. & Roller,P.P. Design and synthesis of novel and potent inhibitors of the type II transmembrane serine protease, matriptase, based upon the sunflower trypsin inhibitor-1 J Med Chem (2007) 50, 5976-5983. 2007 PubMed DOI Design of small-molecule Inhibitors
I12.002 Jiang,S., Li,P., Lee,S.L., Lin,C.Y., Long,Y.Q., Johnson,M.D., Dickson,R.B. & Roller,P.P. Design and synthesis of redox stable analogues of sunflower trypsin inhibitors (SFTI-1) on solid support, potent inhibitors of matriptase Org Lett (2007) 9, 9-12. 2007 PubMed DOI Design of small-molecule Inhibitors
I12.002 Zablotna,E., Jaskiewicz,A., Legowska,A., Miecznikowska,H., Lesner,A. & Rolka,K. Design of serine proteinase inhibitors by combinatorial chemistry using trypsin inhibitor SFTI-1 as a starting structure J Pept Sci (2007) 13, 749-755. 2007 PubMed DOI Design of small-molecule Inhibitors
I12.002 Zablotna,E., Kret,A., Jaskiewicz,A., Olma,A., Leplawy,M.T. & Rolka,K. Introduction of alpha-hydroxymethyamino acid residues in substrate specificity P1 position of trypsin inhibitor SFTI-1 from sunflower seeds retains its activity Biochem Biophys Res Commun (2006) 340, 823-828. 2006 PubMed DOI Mutation, allelic variant or polymorphism
I12.002 Guo,X., Shi,J., Tang,Z., Cui,D. & Zhang,Y. Synthesis and biological activity of seleno sunflower trypsin inhibitor analog Chem Biol Drug Des (2006) 68, 341-344. 2006 PubMed DOI Substrate specificity
Copyright © 2010 by ITB Bari